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(1S,3R)-GNE-502

(1S,3R)-GNE-502

Item no.	HY-132294A-25mg
Manufacturer	MedChem Express
CASRN	1953134-15-0
Amount	25 mg
Category	Reagents & Chemicals Biochemicals
Type	Chemicals
Specific against	other
Citations	[1]Simon Charles Goodacre, et al. Tetrahydro-Pyrido[3,4-b]Indole Estrogen Receptor Modulators And Uses Thereof. WO2016097072A1.
Smiles	C[C@@H]1CC(C2=CC=CC=C2N3)=C3[C@H](C4=CC=C(C=C4)OCCN5CC(C5)CF)N1S(=O)(C)=O
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Available
Product Description	(1S, 3R)-GNE-502 (compound 179) is a potent ERα degrader with an EC50 value of 13 nM against ERα in MCF7 HCS. (1S, 3R)-GNE-502 can be used to research cancer related with estrogen receptor[1].
Shipping	Room temperature
Manufacturers Applications	Cancer-programmed cell death
MolecularWeight	471.59
Clinical_Information	No Development Reported
Manufacturers Research_Area	Cancer
Solubility	10 mM in DMSO
Manufacturers Target	Estrogen Receptor/ERR
Isoform	ERα
Pathway	Vitamin D Related/Nuclear Receptor
Manufacturers Product type	Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 25 mg

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