Comparison

Lu AA33810 European Partner

Item no. HY-107729-100mg
Manufacturer MedChem Express
CASRN 304008-29-5
Amount 100 mg
Quantity options 100 mg 1 ea 5 mg
Category
Type Chemicals
Specific against other
Citations [1]Walker MW, et al. The novel neuropeptide Y Y5 receptor antagonist Lu AA33810 [N-[[trans-4-[(4,5-dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]-methanesulfonamide] exerts anxiolytic- and antidepressant-like effects in rat models of stress sensitivity. J Pharmacol Exp Ther. 2009 Mar;328(3):900-11.
Smiles CS(NC[C@@H](CC1)CC[C@H]1NC2=NC3=C(S2)CCSC4=CC=CC=C34)(=O)=O
ECLASS 10.1 32160000
ECLASS 11.0 32160000
UNSPSC 12000000
Available
Product Description
Lu AA33810 is a potent and selective antagonist of neuropeptide Y5 receptor with a Ki of 1.5 nM for the human receptor. Lu AA33810 exhibts antianxiolytic-like and antidepressant-like effects[1].
Shipping
Room temperature
Manufacturers Applications
Neuroscience-Neuromodulation
MolecularWeight
423.62
Clinical Information
No Development Reported
Manufacturers Research Area
Neurological Disease
Solubility
10 mM in DMSO
Target
Neuropeptide Y Receptor
Manufacturers Target
Neuropeptide Y Receptor
Isoform
NPY Y5 receptor
Manufacturers Pathway
GPCR/G Protein; Neuronal Signaling
Manufacturers Product type
Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 100 mg
Available: In stock
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