Comparison

BTRX-335140 European Partner

Item no. TMO-T14835-25mg
Manufacturer TargetMol
CASRN 2244614-14-8
Amount 25mg
Category
Type Chemicals
Specific against other
Smiles CCc1cc2c(C)c(-c3nc(C)no3)c(N(CC3)CCC3NC3CCOCC3)nc2c(F)c1
ECLASS 10.1 32160000
ECLASS 11.0 32160000
UNSPSC 12000000
Alias Opioid Receptor,Opioid Receptor,Opioid Receptor, CYM-53093
Available
Short Description
BTRX-335140 is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. BTRX-335140 can distribute well into the CNS. ADMET (absorption, distribution, metabolism, excretion, and toxicity) . BTRX-335140 endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats.
Shipping
cool pack
Storage
-20°
Target names or alias
CYM-53093
Molecular Weight
453, 55
Pathway
Neuroscience|||Endocrinology/Hormones|||GPCR/G Protein
Target
Opioid Receptor

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 25mg
Available: In stock
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