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MCH-1 antagonist 1

MCH-1 antagonist 1

Item no.	HY-100331-1ea
Manufacturer	MedChem Express
CASRN	1039825-68-7
Amount	1 ea
Quantity options	100 mg 10mg 1 ea 1mg 5mg
Category	Reagents & Chemicals Biochemicals
Type	Chemicals
Specific against	other
Formula	C25H26N4O2
Citations	[1]Henderson AJ, et al. Tetrahydrocarboline analogs as MCH-1 antagonists. Bioorg Med Chem Lett. 2010 Dec 1;20(23):7024-8.
Smiles	O=C1C=C(OCC2=CC=CC=C2)C=CN1C3=CC4=C(N(CCN5CCCC5)N=C4)C=C3
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Available
Product Description	MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist with a Ki of 2.6 nM. MCH-1 antagonist 1 also inhibits CYP3A4 with an IC50 of 10 μM.
Shipping	Room temperature
Manufacturers Applications	Metabolism-sugar/lipid metabolism
MolecularWeight	414.50
Clinical Information	No Development Reported
Manufacturers Research Area	Metabolic Disease; Endocrinology
Solubility	10 mM in DMSO
Target	Cytochrome P450; MCHR1 (GPR24)
Manufacturers Target	Cytochrome P450; MCHR1 (GPR24)
Isoform	CYP3
Manufacturers Pathway	GPCR/G Protein; Metabolic Enzyme/Protease; Neuronal Signaling
Manufacturers Product type	Reference compound

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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