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P2Y2R/GPR17 antagonist 1

P2Y2R/GPR17 antagonist 1

Item no.	HY-146486-5mg
Manufacturer	MedChem Express
CASRN	2395016-49-4
Amount	5 mg
Specific against	other
Purity	98.85
Citations	[1]Pillaiyar T, et al. Design, synthesis and biological evaluation of suramin-derived dual antagonists of the proinflammatory G protein-coupled receptors P2Y2 and GPR17. Eur J Med Chem. 2020 Jan 15;186:111789.
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Product Description	P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	COVID-19-immunoregulation
MolecularWeight	432.83
Clinical_Information	No Development Reported
Manufacturers Research_Area	Inflammation/Immunology
Solubility	DMSO : 125 mg/mL (ultrasonic)
Manufacturers Target	P2Y Receptor
Isoform	P2Y2 Receptor
Pathway	GPCR/G Protein
Manufacturers Product type	Reference compound

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