Comparison

cay10471-racemate

Item no. V4963-100mg
Manufacturer InvivoChem LLC
CASRN 844639-57-2
Amount 100mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V4963CAS #:844639-57-2Purity >=98%

Description: CAY10471 Racemate (also known as TM-30089 Racemate) is a novel, potent and highly selective prostaglandin D2 receptor CRTH2 antagonist with a Ki of 0.6 nM for hCRTH2, it is selective over human thromboxane A2 receptor TP (Ki, > 10000 nM) or PGD2 receptor DP (Ki, 1200 nM). CAY10471 Racemate also has effect on mouse and rat orthologs of CRTH2. CAY10471 Racemate (Compound 13) inhibits PGD2-induced inositol phosphate or cAMP formation, suppresses beta-arrestin translocation with IC50s of 12 and 3 nM, respectivel

References: J Med Chem. 2005 Feb 24; 48(4):897-900.


CAY10471 Racemate

Molecular Weight: 416.47
Formula: C??H??FN?O?S
CAS No.: 844639-57-2
SMILES: O=C(O)CN1C2=C(C3=C1C=CC=C3)CC(N(S(=O)(C4=CC=C(F)C=C4)=O)C)CC2
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Technical Information
CAY-10471 Racemate; CAY10471 Racemate; CAY 10471 Racemate; TM-30089 Racemate; TM30089 Racemate; TM 30089 Racemate;

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 100mg
Available: In stock
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