Comparison

roluperidone

Item no. V4698-25mg
Manufacturer InvivoChem LLC
CASRN 359625-79-9
Amount 25mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V4698CAS #:359625-79-9Purity >=98%

Description: Roluperidone (formerly also known as CYR-101, MIN-101, CYR101, and MT-210) is a novel and potent cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors with Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively. As a 5-HT2A and sigma 2 receptor antagonist, it can be potentially used for the treatment of schizophrenia.

References: Am J Psychiatry. 2017 Jul 28:appiajp201717010122.


Roluperidone

Name: Roluperidone
CAS#: 359625-79-9
Chemical Formula: C22H23FN2O2
Exact Mass: 366.1744
Molecular Weight: 366.43
Elemental Analysis: C, 72.11; H, 6.33; F, 5.18; N, 7.64; O, 8.73
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Technical Information
Synonym: MT-210; MT 210; MT210; MIN-101; MIN 101; MIN101; CYR-101; CYR 101; CYR101; Roluperidone
IUPAC/Chemical Name: 2-((1-(2-(4-fluorophenyl)-2-oxoethyl)piperidin-4-yl)methyl)isoindolin-1-one
InChi Key: RNRYULFRLCBRQS-UHFFFAOYSA-N
InChi Code: InChI=1S/C22H23FN2O2/c23-19-7-5-17(6-8-19)21(26)15-24-11-9-16(10-12-24)13-25-14-18-3-1-2-4-20(18)22(25)27/h1-8, 16H, 9-15H2
SMILES Code: O=C1N(CC2CCN(CC(C3=CC=C(F)C=C3)=O)CC2)CC4=C1C=CC=C4

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 25mg
Available: In stock
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