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sufugolix

sufugolix

Item no.	V4597-10mg
Manufacturer	InvivoChem LLC
CASRN	308831-61-0
Amount	10mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Description	InvivoChem Cat #:V4597CAS #:308831-61-0Purity >=98% Description: Sufugolix (also known as TAK-013) is a novel, highly potent, non-peptide, selective and orally bioavailable luteinizing hormone-releasing hormone (LHRH) receptor antagonist with an IC50 of 0.1 nM. Sufugolix was under development for the treatment of endometriosis and uterine leiomyoma and reached phase II clinical trials for both of these indications, but was discontinued. References: J Med Chem. 2003 Jan 2; 46(1):113-24.
	Name: Sufugolix CAS#: 308831-61-0 Chemical Formula: C36H31F2N5O4S Exact Mass: 667.2065 Molecular Weight: 667.7318 Elemental Analysis: C, 64.76; H, 4.68; F, 5.69; N, 10.49; O, 9.58; S, 4.80
Storage	-20C for 3 years in powder form
	-80C for 2 years in solvent
Technical Information	Synonym: TAK-013; TAK013; TAK 013. IUPAC/Chemical Name: 1-(4-(5-((benzyl(methyl)amino)methyl)-1-(2, 6-difluorobenzyl)-2, 4-dioxo-3-phenyl-1, 2, 3, 4-tetrahydrothieno[2, 3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea InChi Key: UCQSBGOFELXYIN-UHFFFAOYSA-N InChi Code: InChI=1S/C36H31F2N5O4S/c1-41(20-23-10-5-3-6-11-23)21-28-31-33(44)43(26-12-7-4-8-13-26)36(46)42(22-27-29(37)14-9-15-30(27)38)34(31)48-32(28)24-16-18-25(19-17-24)39-35(45)40-47-2/h3-19H, 20-22H2, 1-2H3, (H2, 39, 40, 45) SMILES Code: O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)CC3=CC=CC=C3)C(C(N4C5=CC=CC=C5)=O)=C2N(CC6=C(F)C=CC=C6F)C4=O)C=C1

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Amount: 10mg

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Delivery expected until 9/6/2024