Comparison

raxatrigine

Item no. V3620-100mg
Manufacturer InvivoChem LLC
CASRN 934240-30-9
Amount 100mg
Category
Type Biochemicals
Specific against other
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Description
InvivoChem Cat #:V3620CAS #:934240-30-9 Purity >=98%

Description: Raxatrigine (also known as GSK1014802 and CNV-1014802) is a novel, potent small molecule state-dependent sodium channel blocker, the Nav1.7 sodium channel inhibitor. It has the potential to be used as an analgesic and is being developed by Convergence Pharmaceuticals for the treatment of lumbosacral radiculopathy (sciatica) and trigeminal neuralgia (TGN).

References: J Pharmacol Exp Ther. 2011 Jul; 338(1):100-13.

Related CAS#: 934240-31-0 (HCl); 934240-30-9 (free base) 934240-35-4 (mesylate)

Raxatrigine
Name: Raxatrigine (GSK1014802)
CAS#: 934240-30-9 (free base).
Chemical Formula: C18H19FN2O2
Exact Mass: 314.14306
Molecular Weight: 314.36
Elemental Analysis: C, 68.77; H, 6.09; F, 6.04; N, 8.91; O, 10.18
Storage
-20C for 3 years in powder form
-80C for 2 years in solvent
Technical Information
Synonym: CNV1014802; CNV-1014802; CNV 1014802; GSK1014802; GSK 1014802; GSK-1014802; Raxatrigine.
Chemical Name: (2S, 5R)-5-(4-((2-fluorobenzyl)oxy)phenyl)pyrrolidine-2-carboxamide
InChi Key: JESCETIFNOFKEU-SJORKVTESA-N
InChi Code: InChI=1S/C18H19FN2O2/c19-15-4-2-1-3-13(15)11-23-14-7-5-12(6-8-14)16-9-10-17(21-16)18(20)22/h1-8, 16-17, 21H, 9-11H2, (H2, 20, 22)/t16-, 17+/m1/s1
SMILES Code: O=C(N)[CH]1N[CH](C2=CC=C(OCC3=CC=CC=C3F)C=C2)CC1

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 100mg
Available: In stock
available

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