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funapide

funapide

Item no.	V21406-250mg
Manufacturer	InvivoChem LLC
CASRN	1259933-16-8
Amount	250mg
Category	Reagents & Chemicals Molecules
Type	Biochemicals
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Description	InvivoChem Cat #:V21406CAS #:1259933-16-8Purity >=98% Description: Funapide (TV-45070; XEN-402) is a novel and potent Sodium Channel Nav1.7 inhibitor, used as an analgesic agent for the treatment of a variety of chronic pain conditions, including osteoarthritis, neuropathic pain, postherpetic neuralgia, and erythromelalgia, as well as dental pain. Funapide acts as a small-molecule Nav1.7 and Nav1.8 voltage-gated sodium channel blocker. References: 1. Safetyand Efficacy of a Topical Sodium Channel Inhibitor (TV-45070) inPatients With Postherpetic Neuralgia (PHN): A Randomized, Controlled, Proof-of-Concept, Crossover Study, With a Subgroup Analysis of theNav1.7 R1150W Genotype. Clin J Pain. 2017 Apr; 33(4):310-318. 2. Recent progressin sodium channel modulators for pain. Bioorg Med Chem Lett. 2014 Aug15; 24(16):3690-9. doi: 10.1016/j.bmcl.2014.06.038. Epub 2014 Jun 21. Review.PubMed PMID: 25060923.

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Amount: 250mg

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