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RET V804M-IN-1

RET V804M-IN-1

Item no.	CS-0130168-10mg
Manufacturer	ChemScene
Amount	10mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Alias	2414909-94-5
Similar products	2414909-94-5
Available
CAS	2414909-94-5
Purity	>98%
MWt	344.37
Formula	C19H16N6O
Solubility	DMSO : 125 mg/mL (362.98 mM; Need ultrasonic)
Clinical Information	No Development Reported
Pathway	Protein Tyrosine Kinase/RTK
Target	RET
Biological Activity	RET V804M-IN-1 (compound 5) is a wt-RET -selective inhibitors of RETV804M kinase, with an IC₅₀ of 20 nM^[1]. IC50 & Target: IC50: 20 nM (RETV804M)^[1]. In Vitro: RET V804M-IN-1 (compound 5) exhibits 3.7 and 110 fold selectivity compared to wt-RET and KDR, respectively^[1].
Research Area	Cancer

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 10mg

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