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WAY-100635 Maleate

WAY-100635 Maleate

Item no.	CS-0019684-5mg
Manufacturer	ChemScene
Amount	5mg
Category	Reagents & Chemicals Molecules
Type	Molecules
Specific against	other
ECLASS 10.1	32169090
ECLASS 11.0	32169090
UNSPSC	12000000
Similar products	1092679-51-0
Available
CAS	1092679-51-0
Purity	>98%
Formula	C29H38N4O6
MWt	538.64
Solubility	H2O : 25 mg/mL (46.41 mM; Need ultrasonic); DMSO : >= 250 mg/mL (464.13 mM)
Clinical Information	No Development Reported
Pathway	Neuronal Signaling; GPCR/G Protein
Target	5-HT Receptor; 5-HT Receptor
Biological Activity	WAY-100635 Maleate is a potent and selective 5-HT_1A Receptor antagonist with a pIC₅₀ of 8.87, an apparent pA₂ of 9.71. IC50 & Target: pIC50 Value: 8.87 (5-HT_1A Receptor)^[1]. In Vitro: WAY-100635 Maleate is a potent and, at high concentrations, an insurmountable antagonist of the 5-HT_1A receptor agonist action of 5-carboxamidotryptamine, with an apparent pA₂ value (at 0.3 nM) of 9.71. WAY-100635 displaces specific binding of the 5-HT_1A radioligand, [³H]8-OH-DPAT (8-hydroxy-2-(di-n-propylamino)tetralin), to rat hippocampal membranes with a plC_IC50 of 8.87^[1].

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 5mg

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