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Chlorprothixene

Chlorprothixene

Item no.	HY-B0274-500mg
Manufacturer	MedChem Express
CASRN	113-59-7
Amount	500 mg
Quantity options	100 mg 10mM/1mL 200 mg 500 mg 50 mg
Category	Food Safety Histamines Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Clone	N/A
Specific against	other
Purity	99.61
Formula	C18H18ClNS
Citations	[1]Y von Coburg, et al. Potential utility of histamine H3 receptor antagonist pharmacophore in antipsychotics. Bioorg Med Chem Lett. 2009 Jan 15;19(2):538-42.<br>[2]B L Roth, et al. Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors. J Pharmacol Exp Ther. 1994 Mar;268(3):1403-10.
Smiles	CN(C)CC/C=C1C2=C(SC3=C\1C=CC=C3)C=CC(Cl)=C2
ECLASS 5.1	30220300
ECLASS 6.1	30220300
ECLASS 8.0	32160605
ECLASS 9.0	32160605
ECLASS 10.0.1	32160490
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	113-59-7
Available
Product Description	Chlorprothixene is a dopamine and histamine receptors antagonist with Kis of 18 nM, 2.96 nM, 4.56 nM, 9 nM and 3.75 nM for hD1, hD2, hD3, hD5 and hH1 receptors, respectively. Antipsychotic activity[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	Neuroscience-Neuromodulation
MolecularWeight	315.86
Clinical_Information	Launched
Manufacturers Research Area	Neurological Disease
Solubility	DMSO : 33.33 mg/mL (ultrasonic)\|H2O : < 0.1 mg/mL
Manufacturers Target	Bacterial; Dopamine Receptor; Histamine Receptor
Isoform	D1 Receptor; D2 Receptor; D3 Receptor; D5 Receptor; H1 Receptor
Pathway	Anti-infection; GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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HY-B0274-500mg-safety-datasheet.pdf