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Bilastine

Bilastine

Item no.	HY-14447-50mg
Manufacturer	MedChem Express
CASRN	202189-78-4
Amount	50 mg
Quantity options	100 mg 10mM/1mL 10 mg 25 mg 50 mg 5 mg
Category	Oncology Food Safety Histamines Inhibitors & Compound Libraries Small Molecules By Organ Skin Cancer Brain Cancer
Type	Inhibitors
Specific against	other
Purity	99.91
Formula	C28H37N3O3
Citations	[1]Corcostegui, R., et al., Preclinical pharmacology of bilastine, a new selective histamine H1 receptor antagonist: receptor selectivity and in vitro antihistaminic activity. Drugs R D, 2005. 6(6): p. 371-84.<br/>[2]Jauregizar, N., et al., Pharmacokinetic-pharmacodynamic modelling of the antihistaminic (H1) effect of bilastine. Clin Pharmacokinet, 2009. 48(8): p. 543-54.
Smiles	CC(C)(C1=CC=C(CCN2CCC(C3=NC4=CC=CC=C4N3CCOCC)CC2)C=C1)C(O)=O
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	202189-78-4
Available
Product Description	Bilastine is a histamine H1 receptor antagonist that can be used to treat allergic rhinoconjunctivitis and urticaria.
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	COVID-19-immunoregulation
MolecularWeight	463.61
Clinical Information	Launched
Manufacturers Research Area	Inflammation/Immunology; Endocrinology
Solubility	DMSO : 10 mg/mL (ultrasonic; warming; heat to 60°C)
Target	Histamine Receptor
Manufacturers Target	Histamine Receptor
Isoform	H1 Receptor
Manufacturers Pathway	GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Manufacturers Product type	Reference compound

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HY-14447-50mg-safety-datasheet.pdf