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(±)-WIN 55,212 (mesylate)

(±)-WIN 55,212 (mesylate)

Item no.	TMO-T38199-50mg
Manufacturer	TargetMol
CASRN	137795-17-6
Amount	50mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitor
Specific against	other
Purity	0,98
Smiles	O=C(C1=CC=CC=2C=CC=CC21)C=3C=4C=CC=C5OCC(N(C54)C3C)CN6CCOCC6.O=S(=O)(O)C
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Short Description	(±)-WIN 55, 212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively. In contrast, the enantiomer (-)-WIN 55, 212-3 acts a partial inverse agonist at CB1 (pIC50 = 5.5) and as a competitive neutral antagonist of CB2, reversing the inverse agonism evoked by SR 144528 (pEC50 = 5.3). (+)-WIN 55, 212 (mesylate) is a mixture of the two enantiomers, (+)-WIN 55, 212-2 and (-)-WIN 55, 212-3.
Shipping	cool pack
Storage	-20°
Molecular Weight	522, 61

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 50mg

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Delivery expected until 9/27/2024

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