MS417

Item no.	TMO-T16154-50mg
Manufacturer	TargetMol
CASRN	916489-36-6
Amount	50mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Purity	99.88%
Citations	Zhang G, et al. Down-regulation of NF-kappaB transcriptional activity in HIV-associated kidney disease by BRD4 inhibition. J Biol Chem. 2012 Aug 17;287(34):28840-51.
Smiles	COC(=O)C[C@@H]1N=C(C2=C(SC(C)=C2C)N2C(C)=NN=C12)C1=CC=C(Cl)C=C1
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	916489-36-6, Epigenetic Reader Domain, GTPL7512
Available
Short Description	MS417 is an inhibitor of BET-specific BRD4(BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weak selectivity at CBP BRD with IC50 of 32.7 μM.
Shipping	cool pack
Storage	-20°
Target names or alias	GTPL7512
Molecular Weight	414, 91
Pathway	Chromatin/Epigenetic\|\|\|Proteases/Proteasome\|\|\|Microbiology/Virology
Target	HIV Protease\|\|\|Epigenetic Reader Domain

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

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Amount: 50mg

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Delivery expected until 8/16/2024

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