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Cyclorasin 9A5

Cyclorasin 9A5

Item no.	HY-P10051
Manufacturer	MedChem Express
CASRN	1782098-79-6
Amount	1 ea
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Formula	C75H108FN25O13
Citations	[1]Koh Takeuchi, et al. Conformational Plasticity of Cyclic Ras-Inhibitor Peptides Defines Cell Permeabilization Activity. Angew Chem Int Ed Engl. 2021 Mar 15;60(12):6567-6572.
Smiles	O=C(N[C@@](C(N[C@@H](C(N[C@H](C(N[C@H](C(N[C@H]1CCCNC(N)=N)=O)CCCNC(N)=N)=O)CCCNC(N)=N)=O)C)=O)([H])[C@H](O)C)[C@@H](NC([C@@H](NC([C@H](NC([C@@H](NC([C@@H](NC([C@H](NC1=O)CC2=CC(C=CC=C3)=C3C=C2)=O)CCCNC(N)=N)=O)CC(C=C4)=CC=C4F)=O)CCCC)=O)CCC(N)=O)=O)CC5=CNC6=CC=CC=C56
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Product Description	Cyclorasin 9A5 is an 11-residue cell-permeable cyclic peptide that orthosterically inhibits the Ras-Raf protein interaction with an IC50 of 120 nM[1].
Shipping	Room temperature
Manufacturers Applications	Cancer-Kinase/protease
MolecularWeight	1586.82
Clinical Information	No Development Reported
Manufacturers Research Area	Cancer
Solubility	10 mM in DMSO
Target	Raf; Ras
Manufacturers Target	Raf; Ras
Manufacturers Pathway	GPCR/G Protein; MAPK/ERK Pathway
Manufacturers Product type	Peptides

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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