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Lemborexant

Lemborexant

Item no.	HY-16725-100mg
Manufacturer	MedChem Express
CASRN	1369764-02-2
Amount	100 mg
Quantity options	100 mg 10 mM x 1 mL 10 mg 25 mg 50 mg 5 mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitor
Specific against	other
Purity	99.19%
Citations	bioRxiv. 2020 May.
Smiles	O=C([C@H]1[C@@](C2=CC=CC(F)=C2)(COC3=CN=C(C)N=C3C)C1)NC4=NC=C(F)C=C4
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	E-2006
Available
Product Description	Lemborexant (E-2006) is a reversible, competitive and orally active dual antagonist of the orexin OX1 and OX2 receptors with IC50 values of 6.1 nM and 2.6 nM, respectively. Lemborexant can be treated insomnia.
StorageTemperature	Powder -20°C 3 years, 4°C 2 years; In solvent -80°C 6 months, -20°C 1 month
MolecularWeight	410.42
Clinical_Information	Launched
Research_Area	Neurological Disease
Solubility	DMSO : 100 mg/mL (243.65 mM; Need ultrasonic)
Target	Orexin Receptor (OX Receptor)
Isoform	OX1; OX2
Pathway	GPCR/G Protein; Neuronal Signaling

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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