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Timapiprant (sodium)

Timapiprant (sodium)

Manufacturer	MedChem Express
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Amount	100 mg
Item no.	HY-15342A-100mg
CASRN	950688-14-9
eClass 6.1	30220300
eClass 9.0	32160605
Available
Alias	OC000459 (sodium)
Purity	99.61
Product Description	Timapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. Timapiprant sodium (OC000459 sodium) potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), and human native DP2 (Ki=4 nM). Timapiprant sodium (OC000459 sodium) inhibits mast cell activation of Th2 lymphocytes and eosinophils[1].
StorageTemperature	4°C (Powder, stored under nitrogen)
Shipping	Room Temperature
Manufacturers Applications	Neuroscience-Neuromodulation
MolecularWeight	370.35
Clinical_Information	Phase 2
Manufacturers Research_Area	Inflammation/Immunology; Endocrinology
Solubility	DMSO : 100 mg/mL (ultrasonic)
Manufacturers Target	Prostaglandin Receptor
Isoform	DP
Pathway	GPCR/G Protein
Manufacturers Product type	Reference compound

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