Comparison

CB2R/FAAH modulator-2 European Partner

Item no. HY-152253-5mg
Manufacturer MedChem Express
CASRN 2876918-68-0
Amount 5 mg
Category
Type Inhibitors
Specific against other
Purity 99.59
Formula C24H33NO2
Citations [1]Francesca Intranuovo, et al. Development of N-(1-Adamantyl)benzamides as Novel Anti-Inflammatory Multitarget Agents Acting as Dual Modulators of the Cannabinoid CB2 Receptor and Fatty Acid Amide Hydrolase. J Med Chem. 2023 Jan 12;66(1):235-250.
Smiles O=C(C1=C(OCC2CCCCC2)C=CC=C1)NC3(C4)C[C@H]5C[C@@H]4C[C@H](C5)C3
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Available
Product Description
CB2R/FAAH modulator-2 (compound 26) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-2 are 10.8 and 152.9 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 6.2 μM. CB2R/FAAH modulator-2 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection[1].
StorageTemperature
-20°C, 3 years; 4°C, 2 years (Powder)
Shipping
Room Temperature
Manufacturers Applications
COVID-19-anti-virus
MolecularWeight
367.52
Clinical_Information
No Development Reported
Manufacturers Research_Area
Cancer; Infection; Inflammation/Immunology; Neurological Disease
Solubility
10 mM in DMSO
Manufacturers Target
Cannabinoid Receptor; FAAH
Isoform
CB1; CB2
Pathway
GPCR/G Protein; Metabolic Enzyme/Protease; Neuronal Signaling
Manufacturers Product type
Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 5 mg
Available: In stock
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