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Bromodomain IN-2

Bromodomain IN-2

Item no.	HY-149806-1ea
Manufacturer	MedChem Express
CASRN	2445335-77-1
Amount	1 ea
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Formula	C16H17ClN2O
Citations	[1]Warstat R, et al. A novel pan-selective bromodomain inhibitor for epigenetic drug design. Eur J Med Chem. 2023 Mar 5;249:115139.
Smiles	O=C1C2=C(C)NC(C3=C(Cl)C=CC(N)=C3)=C2CCCC1
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Product Description	Bromodomain IN-2 is a pan bromodomain (BD) inhibitor with KD values of 250, 420, 130, 430, 67, 240, 970 nM for BRD4(1), CBP, BRPF1B, BRD7, BRD9, BRDT(1), CECR2 respectively. Bromodomain IN-2 shows antiproliferative activity[1].
Shipping	Room temperature
Manufacturers Applications	Cancer-programmed cell death
MolecularWeight	288.77
Clinical Information	No Development Reported
Manufacturers Research Area	Cancer
Solubility	10 mM in DMSO
Target	Epigenetic Reader Domain
Manufacturers Target	Epigenetic Reader Domain
Isoform	BRD4; BRD7; BRD9; BRDT; BRPF1
Manufacturers Pathway	Epigenetics
Manufacturers Product type	Reference compound

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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