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PCAF-IN-2

PCAF-IN-2

Item no.	HY-147895-25mg
Manufacturer	MedChem Express
CASRN	56173-05-8
Amount	25 mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitor
Specific against	other
Purity	98.0
Formula	C10H7F3N6
Citations	[1]Turky A, et al. Design, synthesis, and antitumor activity of novel compounds based on 1,2,4-triazolophthalazine scaffold: Apoptosis-inductive and PCAF-inhibitory effects. Bioorg Chem. 2020 Aug;101:104019.
Smiles	FC(C1=NN=C2N1N=C(NN)C3=C2C=CC=C3)(F)F
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Product Description	PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phase[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	Cancer-programmed cell death
MolecularWeight	268.20
Clinical_Information	No Development Reported
Manufacturers Research_Area	Cancer
Solubility	DMSO : 8.33 mg/mL (ultrasonic; warming; heat to 80°C)
Manufacturers Target	Apoptosis; Histone Acetyltransferase
Isoform	GCN5/PCAF
Pathway	Apoptosis; Epigenetics
Manufacturers Product type	Reference compound

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