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CCR2 antagonist 1

CCR2 antagonist 1

Item no.	HY-112792-10mM
Manufacturer	MedChem Express
CASRN	1683534-96-4
Amount	10mM/1mL
Quantity options	10mM/1mL 10 mg 1 mg 50 mg 5 mg
Category	Metabolism Cholesterol & Lipid Metabolism Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Purity	98.00
Formula	C28H32BrF3N2O
Citations	[1]Vilums M, et al. When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists. Eur J Med Chem. 2015 Mar 26;93:121-34.
Smiles	O=C([C@]1(C(C)C)C[C@H](N[C@@H]2CCC3=C2C=CC(Br)=C3)CC1)N4CC5=C(C=CC(C(F)(F)F)=C5)CC4
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	1683534-96-4
Similar products	1683534-96-4
Available
Product Description	CCR2 antagonist 1 (compound 15a) is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	Metabolism-protein/nucleotide metabolism
MolecularWeight	549.47
Clinical Information	No Development Reported
Manufacturers Research Area	Endocrinology
Solubility	DMSO : 125 mg/mL (ultrasonic)
Target	CCR
Manufacturers Target	CCR
Isoform	CCR2
Manufacturers Pathway	GPCR/G Protein; Immunology/Inflammation
Manufacturers Product type	Reference compound

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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