MT1

Item no.	HY-111976-10mM
Manufacturer	MedChem Express
CASRN	2060573-82-0
Amount	10mM/1mL
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitor
Specific against	other
Purity	99.78
Formula	C54H66Cl2N10O9S2
Citations	[1]Minoru Tanaka, et al. Design and characterization of bivalent BET inhibitors. Nat Chem Biol. 2016 Dec;12(12):1089-1096.
Smiles	CC1=NN=C2N1C3=C(C(C4=CC=C(C=C4)Cl)=N[C@H]2CC(NCCOCCOCCOCCOCCOCCOCCOCCNC(C[C@@H]5N=C(C6=C(N7C5=NN=C7C)SC(C)=C6C)C8=CC=C(C=C8)Cl)=O)=O)C(C)=C(C)S3
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Product Description	MT1 is a bivalent chemical probe of BET bromodomains, with an IC50 of 0.789 nM for BRD4(1)[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	Cancer-programmed cell death
MolecularWeight	1134.20
Clinical_Information	No Development Reported
Manufacturers Research_Area	Cancer
Solubility	DMSO : 150 mg/mL (ultrasonic)
Manufacturers Target	Epigenetic Reader Domain
Pathway	Epigenetics
Manufacturers Product type	Reference compound

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