Comparison

CDK9-IN-8 European Partner

Item no. HY-102039-5mg
Manufacturer MedChem Express
CASRN 2105956-51-0
Amount 5 mg
Quantity options 100 mg 10 mg 1 mg 25 mg 50 mg 5 mg
Category
Type Inhibitors
Specific against other
Purity 99.65
Formula C31H32FN7O3
Citations [1]Li Y, et al. Discovery of a highly potent, selective and novel CDK9 inhibitor as an anticancer drug candidate. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3231-3237.
Smiles FC1=CC=C(NC(C2(CC2)C(NC3=CC=C(NC4=NC=C5C(N(C6CCCC6)C(C(N(C)C)=O)=C5)=N4)C=C3)=O)=O)C=C1
ECLASS 10.1 32160490
ECLASS 11.0 32160490
UNSPSC 12000000
Alias 2105956-51-0
Available
Product Description
CDK9-IN-8 is a highly effective and selective CDK9 inhibitor with an IC50 of 12 nM.
StorageTemperature
-20°C, 3 years; 4°C, 2 years (Powder)
Shipping
Room Temperature
Manufacturers Applications
Cancer-Kinase/protease
MolecularWeight
569.63
Clinical Information
No Development Reported
Manufacturers Research Area
Cancer
Solubility
DMSO : 5.2 mg/mL (ultrasonic; warming; heat to 80°C)|H2O : 1 mg/mL (ultrasonic; warming; heat to 80°C)
Target
CDK
Manufacturers Target
CDK
Isoform
CDK9
Manufacturers Pathway
Cell Cycle/DNA Damage
Manufacturers Product type
Reference compound

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

Amount: 5 mg
Available: In stock
available

Compare

Add to wishlist

Get an offer

Request delivery time

Ask a technical question

Submit a bulk request

Questions about this Product?
 
Close