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MCHR1 antagonist 2

MCHR1 antagonist 2

Item no.	HY-100321-25mg
Manufacturer	MedChem Express
CASRN	863115-70-2
Amount	25 mg
Quantity options	100 mg 10 mM/1mL 10 mg 1 mg 25 mg 50 mg 5 mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Purity	98.27
Formula	C23H21FN2O5
Citations	[1]Lynch JK, et al. Optimization of chromone-2-carboxamide melanin concentrating hormone receptor 1 antagonists: assessment of potency, efficacy, and cardiovascular safety. J Med Chem. 2006 Nov 2;49(22):6569-84.
Smiles	O=C(C1=CC(C2=CC(F)=CC=C2O1)=O)NC3CCN(CC4=CC=C(OCO5)C5=C4)CC3
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	863115-70-2
Similar products	863115-70-2
Available
Product Description	MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells[1].
StorageTemperature	-20°C, 3 years; 4°C, 2 years (Powder)
Shipping	Room Temperature
Manufacturers Applications	Metabolism-protein/nucleotide metabolism
MolecularWeight	424.42
Clinical Information	No Development Reported
Manufacturers Research Area	Metabolic Disease; Endocrinology
Solubility	DMSO : 10 mg/mL (ultrasonic; adjust pH to 6 with HCl)
Target	MCHR1 (GPR24); Potassium Channel
Manufacturers Target	MCHR1 (GPR24); Potassium Channel
Manufacturers Pathway	GPCR/G Protein; Membrane Transporter/Ion Channel; Neuronal Signaling
Manufacturers Product type	Reference compound

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