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TG101209

TG101209

Item no.	DCC-DC7317-10mM
Manufacturer	DCChemicals
CASRN	936091-14-4
Amount	10 mM x 1 mL in DMSO
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
Smiles	C(S(NC(C)(C)C)(=O)=O)1=CC=CC(NC2C(C)=CN=C(NC3=CC=C(N4CCN(C)CC4)C=C3)N=2)=C1
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Available
Molecule Weight	509, 67
Field of Application	TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM, less potent to Flt3 and RET with IC50 of 25 nM and 17 nM, ~30-fold selective for JAK2 than JAK3, sensitive to JAK2V617F and MPLW515L/K mutations; TG101209 inhibit BRD4 activity with IC50 of 130 nM.

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 10 mM x 1 mL in DMSO

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Delivery expected until 9/6/2024

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