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CNT2 inhibitor-1

CNT2 inhibitor-1

Item no.	CS-0066911-100mg
Manufacturer	ChemScene
Amount	100mg
Category	Inhibitors & Compound Libraries Small Molecules
Type	Inhibitors
Specific against	other
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Similar products	880155-70-4
Available
CAS	880155-70-4
Purity	>98%
Formula	C23H24N6O4
MWt	448.47
Solubility	DMSO : 75 mg/mL (167.24 mM; Need ultrasonic)
Clinical Information	No Development Reported
Pathway	Others
Target	Others
Biological Activity	CNT2 inhibitor-1 is a potent concentrative nucleoside transporter 2 Inhibitor (CNT2), with an IC₅₀ of 640 nM for hCNT2. IC50 & Target: IC50: 640 nM (hCNT2)^[1]^[2]. In Vitro: CNT2 inhibitor-1 (compound 48) exhibits 81-fold more potent inhibitory activity than the parent compound 12. In addition, CNT2 inhibitor-1 exhibits inhibitory activity 1500-fold more potent than that of 2ï¿½-deoxy-5-fluorouridine, phlorizin, and 7, 8, 3ï¿½-trihydroxyflavone, which are well-known hCNT2 inhibitors^[1]. CNT2 inhibitor-1 (compound 1) is a potent inhibitor with poor solubility^[2].

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All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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