Tacrolimus

ArtNr	HY-13756-100mg
Hersteller	MedChem Express
CAS-Nr.	104987-11-3
Menge	100 mg
Quantity options	100 mg 10 mg 200 mg 500 mg 50 mg 5 mg
Kategorie	Food Safety Drugs Histamines Hormones Neuroscience Metabolism Cholesterol & Lipid Metabolism Neural Signaling Enzymes Other Fatty Acid Enzymes Inhibitors & Compound Libraries Small Molecules
Typ	Inhibitors
Clon	N/A
Specific against	other
Purity	99.93
Formula	C44H69NO12
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Smiles	O=C([C@@](CCCC1)([H])N1C(C([C@@]2(O)[C@H](C)C[C@H](OC)[C@@](O2)([H])[C@@H](OC)C[C@@H](C)C/C(C)=C/[C@H]3CC=C)=O)=O)O[C@H](/C(C)=C/[C@H]4C[C@@H](OC)[C@H](O)CC4)[C@H](C)[C@@H](O)CC3=O
ECLASS 10.1	32160490
ECLASS 11.0	32160490
UNSPSC	12000000
Alias	FK506; Fujimycin; FR900506
Lieferbar
Product Description	Tacrolimus (FK506), a macrocyclic lactone, binds to FK506 binding protein (FKBP) to form a complex. Tacrolimus inhibits calcineurin phosphatase, which inhibits T-lymphocyte signal transduction and IL-2 transcription. Immunosuppressive properties[1].
StorageTemperature	4°C (Powder, protect from light)
Shipping	Room Temperature
Manufacturers Applications	COVID-19-immunoregulation
MolecularWeight	804.02
Clinical Information	Launched
Manufacturers Research Area	Cancer; Infection; Inflammation/Immunology
Solubility	DMSO : ≥ 150 mg/mL
Target	Antibiotic; Autophagy; Bacterial; FKBP; Phosphatase
Manufacturers Target	Antibiotic; Autophagy; Bacterial; FKBP; Phosphatase
Isoform	Macrolide
Manufacturers Pathway	Anti-infection; Apoptosis; Autophagy; Immunology/Inflammation; Metabolic Enzyme/Protease
Manufacturers Product type	Natural Products

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HY-13756-100mg-safety-datasheet.pdf